Deprecated: The each() function is deprecated. This message will be suppressed on further calls in /home/zhenxiangba/zhenxiangba.com/public_html/phproxy-improved-master/index.php on line 456
NZ773357B2 - Systems and methods for producing synthetic hypericin - Google Patents
[go: Go Back, main page]

NZ773357B2 - Systems and methods for producing synthetic hypericin - Google Patents

Systems and methods for producing synthetic hypericin Download PDF

Info

Publication number
NZ773357B2
NZ773357B2 NZ773357A NZ77335716A NZ773357B2 NZ 773357 B2 NZ773357 B2 NZ 773357B2 NZ 773357 A NZ773357 A NZ 773357A NZ 77335716 A NZ77335716 A NZ 77335716A NZ 773357 B2 NZ773357 B2 NZ 773357B2
Authority
NZ
New Zealand
Prior art keywords
hypericin
bicarbonate
precipitation temperature
methods
photoconverting
Prior art date
Application number
NZ773357A
Other versions
NZ773357A (en
Inventor
Rasappa Arumugham
Holger Rauter
Christopher Schaber
Silvia Werner
Original Assignee
Soligenix Inc
Filing date
Publication date
Application filed by Soligenix Inc filed Critical Soligenix Inc
Priority to NZ773357A priority Critical patent/NZ773357B2/en
Priority claimed from PCT/US2016/020189 external-priority patent/WO2017151111A1/en
Publication of NZ773357A publication Critical patent/NZ773357A/en
Publication of NZ773357B2 publication Critical patent/NZ773357B2/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00Systems containing at least three condensed rings
    • C07C2603/02Ortho- or ortho- and peri-condensed systems
    • C07C2603/54Ortho- or ortho- and peri-condensed systems containing more than five condensed rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C46/00Preparation of quinones
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C46/00Preparation of quinones
    • C07C46/10Separation; Purification; Stabilisation; Use of additives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C50/00Quinones
    • C07C50/26Quinones containing groups having oxygen atoms singly bound to carbon atoms
    • C07C50/36Quinones containing groups having oxygen atoms singly bound to carbon atoms the quinoid structure being part of a condensed ring system having four or more rings

Abstract

Improved systems and methods for producing synthetic hypericin at high volume and high purity.

Claims (4)

What is claimed is:
1. A method of preparing a purified synthetic hypericin, the method comprising: (a) photoconverting protohypericin to crude hypericin using a continuous flow micro-reactor; (b) treating the crude hypericin with at least one salt forming reagent in a solvent at a pre- precipitation temperature wherein the at least one salt forming reagent is selected from the group consisting of sodium bicarbonate, ammonium bicarbonate, potassium bicarbonate, calcium bicarbonate, and magnesium bicarbonate; (c) filtering the treated hypericin from step (b) while simultaneously providing at least one cooling ramp in a double jacketed glass vessel equipped with a heating and cooling system to reach a post- precipitation temperature, wherein a precipitate is formed; (d) washing and filtering the precipitate from step (c) with a washing solvent; and (e) drying of the product of step (d) with nitrogen or water vapor, wherein the synthetic hypericin is a mono-sodium salt in the form of a trihydrate at a yield of at least 75% to 100% of the dry product.
2. The method of claim 1, wherein the photoconverting is the result of exposure to a LED light at a wavelength between 350-700 nm.
3. The method of claim 1 or claim 2, wherein pre-precipitation temperature is greater than 40 °C.
4. The method of any one of claims 1 to 3, wherein the post-precipitation temperature is less than 40 °C.
NZ773357A 2016-03-01 Systems and methods for producing synthetic hypericin NZ773357B2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
NZ773357A NZ773357B2 (en) 2016-03-01 Systems and methods for producing synthetic hypericin

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
NZ773357A NZ773357B2 (en) 2016-03-01 Systems and methods for producing synthetic hypericin
PCT/US2016/020189 WO2017151111A1 (en) 2016-03-01 2016-03-01 Systems and methods for producing synthetic hypericin
NZ746762A NZ746762B2 (en) 2016-03-01 Systems and methods for producing synthetic hypericin

Publications (2)

Publication Number Publication Date
NZ773357A NZ773357A (en) 2024-07-26
NZ773357B2 true NZ773357B2 (en) 2024-10-30

Family

ID=

Similar Documents

Publication Publication Date Title
Choi Thermal type seawater desalination with barometric vacuum and solar energy
MY191517A (en) A clean method for preparing d, l-methionine
US10442766B1 (en) Method and production line for preparing 2,6-dichloropyridine through gas phase photochlorination of pyridine
MY188994A (en) A method of producing a two-dimensional material
CL2025000655A1 (en) System and method for magma-driven thermochemical processes
JP2013503913A5 (en)
WO2016023884A3 (en) Method for in-situ regeneration of activated carbon loaded with trihalomethanes using alkaline hydrolysis
NZ773357B2 (en) Systems and methods for producing synthetic hypericin
NZ773357A (en) Systems and methods for producing synthetic hypericin
AR081267A1 (en) PROCEDURE FOR OBTAINING THE CRYSTAL FORM A OF FEBUXOSTAT
Li et al. Two new diphenylethylenes from Arundina graminifolia and their cytotoxicity
RU2018138147A (en) METHOD FOR PRODUCING 5- (BROMMETHYL) -1-BENZOTIOPHENE
WO2017125496A3 (en) Improved method for processing magnesium chloride solutions and method for manufacturing carboxylic acids
RU2017123052A (en) METHOD FOR PRODUCING CARBONIC ACID ANHYDRIDE
MX2016002733A (en) SYNTHESIS PROCESS FOR THE OBTAINING OF USEFUL QUATERNARY CATION SALES AS CHEMICAL DRAWERS IN CARBONATED ROADS, AND PRODUCTS OBTAINED WITH THE SAME.
HRP20140255T1 (en) Method for producing phosphates and compounds containing phosphates, in particular alkaline-earth phosphates, alkaline-earth silicophosphates or alkaline-earth oxides
CN101244829A (en) Thermal treatment of soda mother liquor and production of ammonium chloride industrial technology
US11634338B1 (en) Process for producing aluminum chlorohydrate particles
WO2019132663A8 (en) Method for purifying and removing color of fdca
WO2016055456A3 (en) Production of an aromatic dicarboxylic acid
BR112013006715A2 (en) process and system
WO2016105107A3 (en) Efficient method for producing and purifying anhydrous sugar alcohol
EA201792523A1 (en) METHOD AND SYSTEM OF THERMAL TREATMENT OF GRANULAR SOLID SUBSTANCES
MY185113A (en) Production method of ?-olefin oligomer
CN104446356B (en) Shale hangs the preparation method of picture