AU631433B2 - Synthesis of aryl substituted halohydrins - Google Patents

Synthesis of aryl substituted halohydrins

Info

Publication number: AU631433B2
Authority: AU; Australia
Prior art keywords: halohydrins; synthesis; aryl substituted; aryl; substituted
Prior art date: 1985-12-04
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Ceased

Application number

AU57562/90A

Other versions

AU5756290A (en

Inventor

Khuong H.X. Mai

William L. Matier

Ghanshyam Patil

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Bristol Myers Squibb Pharma Co

Original Assignee

DuPont Merck Pharmaceutical Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1985-12-04

Filing date

1990-06-18

Publication date

1992-11-26

1990-06-18 Application filed by DuPont Merck Pharmaceutical Co filed Critical DuPont Merck Pharmaceutical Co

1990-10-11 Publication of AU5756290A publication Critical patent/AU5756290A/en

1992-06-04 Assigned to DU PONT MERCK PHARMACEUTICAL COMPANY, THE reassignment DU PONT MERCK PHARMACEUTICAL COMPANY, THE Alteration of Name(s) of Applicant(s) under S113 Assignors: E.I. DU PONT DE NEMOURS AND COMPANY

1992-11-26 Application granted granted Critical

1992-11-26 Publication of AU631433B2 publication Critical patent/AU631433B2/en

2006-11-14 Anticipated expiration legal-status Critical

Status Ceased legal-status Critical Current

Links

125000003118 aryl group Chemical group 0.000 title 1
230000015572 biosynthetic process Effects 0.000 title 1
150000003944 halohydrins Chemical class 0.000 title 1
238000003786 synthesis reaction Methods 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
- C07D285/01—Five-membered rings
- C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
- C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
- C07D285/10—1,2,5-Thiadiazoles; Hydrogenated 1,2,5-thiadiazoles
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C41/00—Preparation of ethers; Preparation of compounds having groups, groups or groups
- C07C41/01—Preparation of ethers
- C07C41/18—Preparation of ethers by reactions not forming ether-oxygen bonds
- C07C41/22—Preparation of ethers by reactions not forming ether-oxygen bonds by introduction of halogens; by substitution of halogen atoms by other halogen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
- C07D303/02—Compounds containing oxirane rings
- C07D303/12—Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms
- C07D303/18—Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms by etherified hydroxyl radicals
- C07D303/20—Ethers with hydroxy compounds containing no oxirane rings
- C07D303/22—Ethers with hydroxy compounds containing no oxirane rings with monohydroxy compounds
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Chemical Kinetics & Catalysis (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
Furan Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Indole Compounds (AREA)
Epoxy Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

AU57562/90A 1985-12-04 1990-06-18 Synthesis of aryl substituted halohydrins Ceased AU631433B2 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US80440685A	1985-12-04	1985-12-04
US804406		1985-12-04

Related Parent Applications (1)

Application Number	Title	Priority Date	Filing Date
AU67749/87A Division AU604005B2 (en)	1985-12-04	1986-11-14	Synthesis of aryloxypropanolamines and arylethanolamines

Publications (2)

Publication Number	Publication Date
AU5756290A AU5756290A (en)	1990-10-11
AU631433B2 true AU631433B2 (en)	1992-11-26

Family

ID=25188898

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
AU67749/87A Ceased AU604005B2 (en)	1985-12-04	1986-11-14	Synthesis of aryloxypropanolamines and arylethanolamines
AU57562/90A Ceased AU631433B2 (en)	1985-12-04	1990-06-18	Synthesis of aryl substituted halohydrins

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
AU67749/87A Ceased AU604005B2 (en)	1985-12-04	1986-11-14	Synthesis of aryloxypropanolamines and arylethanolamines

Country Status (6)

Country	Link
EP (1)	EP0248879A4 (en)
JP (1)	JPS63502585A (en)
AU (2)	AU604005B2 (en)
CA (1)	CA1282787C (en)
WO (1)	WO1987003583A1 (en)
ZA (1)	ZA868713B (en)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4990668A (en) *	1985-12-04	1991-02-05	E. I. Du Pont De Nemours And Company	Optically active aryloxypropanolamines and arylethanolamines
SE8801518D0 (en) *	1988-04-22	1988-04-22	Astra Pharma Prod	A NOVEL PROCESS
US4992535A (en) *	1988-10-26	1991-02-12	G. D. Searle & Co.	Methods of making novel R and S diastereomers of N6 -[(2-hydroxypropyl)aryl]adenosines
US5030624A (en) *	1988-10-26	1991-07-09	G. D. Searle & Co.	R-diastereomer of an N6 -[(2-hydroxypropyl)aryl]adenosine and its medicinal uses
US5032584A (en) *	1988-10-26	1991-07-16	G. D. Searle & Co.	S-diastereomer of an n6 -((2-hydroxypropyl)aryl)adenosine and its medicinal uses
DE3844410A1 (en) *	1988-12-30	1990-07-19	Lindner Wolfgang	Inversion of the alcohol configuration in alpha-amino alcohols via intramolecular substitution of the sulphonate groups
US5629345A (en) *	1993-07-23	1997-05-13	Vide Pharmaceuticals	Methods and compositions for ATP-sensitive K+ channel inhibition for lowering intraocular pressure
US5965620A (en) *	1993-07-23	1999-10-12	Vide Pharmaceuticals	Methods and compositions for ATP-sensitive K+ channel inhibition for lowering intraocular pressure
AR011626A1 (en) *	1997-02-07	2000-08-30	Shell Int Research	A PROCEDURE FOR THE ELABORATION OF EPOXID COMPOUNDS, EPOXID RESINS OBTAINED THROUGH SUCH A PROCEDURE AND A PROCEDURE FOR THE ELABORATION OF INTERMEDIATE COMPOUNDS FOR THE ELABORATION OF EPOXID COMPOUNDS
BR112013018598A2 (en) *	2011-01-27	2016-10-18	Baxter Healthcare Sa	pharmaceutical composition, method for treating heart disease, use of (s) -methyl-3- [4- (2-hydroxy-3- [4- (2-hydroxy-3-isopropylamino) propoxy] phenylpropionate, and method for control heart rate
JP2014505074A (en) *	2011-01-27	2014-02-27	バクスター・インターナショナル・インコーポレイテッド	Method for treating tachycardia and / or controlling heart rate while minimizing and / or controlling hypotension
CN102408285B (en) *	2011-09-15	2013-11-20	东北师范大学	Method for directly aminating benzyl hydrocarbon of methylbenzene derivative

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4202978A (en) *	1978-02-08	1980-05-13	Hoffmann-La Roche Inc.	(S)-1-[2-(4-(2-Hydroxy-s-(1-alkylaminopropoxy)phenylalkyl]-4-phenylpiperazines
US4990668A (en) *	1985-12-04	1991-02-05	E. I. Du Pont De Nemours And Company	Optically active aryloxypropanolamines and arylethanolamines

1986
- 1986-11-14 EP EP19870900373 patent/EP0248879A4/en not_active Withdrawn
- 1986-11-14 CA CA000522978A patent/CA1282787C/en not_active Expired - Lifetime
- 1986-11-14 AU AU67749/87A patent/AU604005B2/en not_active Ceased
- 1986-11-14 WO PCT/US1986/002406 patent/WO1987003583A1/en not_active Ceased
- 1986-11-14 JP JP62500136A patent/JPS63502585A/en active Pending
- 1986-11-17 ZA ZA868713A patent/ZA868713B/en unknown
1990
- 1990-06-18 AU AU57562/90A patent/AU631433B2/en not_active Ceased

Also Published As

Publication number	Publication date
JPS63502585A (en)	1988-09-29
EP0248879A4 (en)	1990-02-26
CA1282787C (en)	1991-04-09
AU5756290A (en)	1990-10-11
AU6774987A (en)	1987-06-30
ZA868713B (en)	1987-06-24
EP0248879A1 (en)	1987-12-16
AU604005B2 (en)	1990-12-06
WO1987003583A1 (en)	1987-06-18

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EP0196078A3 (en)	1987-04-15	Synthesis of improved zeolites
AU631433B2 (en)	1992-11-26	Synthesis of aryl substituted halohydrins
AU2075388A (en)	1989-01-19	Novel synthesis of 3-amino-2-methylbenzotrifluoride
GB8612528D0 (en)	1986-07-02	Synthesis of zsm-23
AU568706B2 (en)	1988-01-07	Synthesis of silicophosphoaluminates
AU573085B2 (en)	1988-05-26	Production of monotertiarybutyl toluinediamines
AU583297B2 (en)	1989-04-27	Improved synthesis of ZSM-23 zeolite
EG17986A (en)	1991-08-30	Synthesis of tricyclazole
AU582932B2 (en)	1989-04-13	Synthesis of nizatidine
AU4886885A (en)	1986-04-24	Synthesis of quinones
JPS6490139A (en)	1989-04-06	Synthesis of cis-9-tricocene
AU575985B2 (en)	1988-08-11	Synthesis of silicophosphoaluminate
AU6842587A (en)	1987-08-14	Prostaglandin synthesis
AU8827382A (en)	1984-02-08	Synthesis of periplanone-b
AU587847B2 (en)	1989-08-31	Manufacture of hydrocarbons
AU589631B2 (en)	1989-10-19	Purification of 5-pyrimidinecarboxamides
GB8416903D0 (en)	1984-08-08	Synthesis of clavulone derivatives
IE850075L (en)	1985-07-12	Synthesis of aminonitropyridines.
GB8431904D0 (en)	1985-01-30	Synthesis of yeuhchukene
IE851525L (en)	1986-01-11	Synthesis of 1,3-dioxanes