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AU653619B2 - Medicament against cancer and AIDS - Google Patents
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AU653619B2 - Medicament against cancer and AIDS - Google Patents

Medicament against cancer and AIDS Download PDF

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Publication number
AU653619B2
AU653619B2 AU21253/92A AU2125392A AU653619B2 AU 653619 B2 AU653619 B2 AU 653619B2 AU 21253/92 A AU21253/92 A AU 21253/92A AU 2125392 A AU2125392 A AU 2125392A AU 653619 B2 AU653619 B2 AU 653619B2
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AU
Australia
Prior art keywords
aids
nadh
treatment
therapy
nadph
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Ceased
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AU21253/92A
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AU2125392A (en
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Jorg Univ.-Prof. DDR. Birkmayer
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Virology (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Molecular Biology (AREA)
  • Epidemiology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • AIDS & HIV (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Saccharide Compounds (AREA)

Abstract

Use of nicotinamide adenine dinucleotide (NADH), nicotinamide adenine dinucleotide phosphate (NADPH) or of a physiologically tolerated salt thereof for the treatment of cancer or AIDS.

Description

P100/011 2815101 Regulation 3.2(2)
AUSTRALIA
Patents Act 1990 653619
ORIGINAL
COMPLETE SPECIFICATION STANDARD PATENT Application Number: Lodged: Invention Title: MEDICAMENT AGINST CANCER AND AIDS The following statement Is a full description of this lnven:n, Including the best method of performing It known to :-ME Medicament against cancer Ov AIDS.
The invention relates to the novel use of nicotinamide-adenine dinucleotide (NADH), nicotinamide-adenine dinucleotide phosphate (NADPH) or a physiologically compatible salt thereof.
Cancer has numerous different manifestations and the genesis thereof is in many cases not yet completely clarified and, apart from genetic predispositions, as a function of the tumour type certain risk factors would appear to play a part. The therapy of cancer is essentially based on operating, radiotherapy and chemotherapy, which are often used in combination and have different success rates as a function of the tumour type. Each of these therapy forms represents a severe course of action with all the associated risks and side effects.
S* Acquired immune deficiency syndrome or AIDS described as a separate disease for the first time in 1981 is characterized by persistent or recurrent diseases which only occur in the advanced stage thereof and Swhich indicate defects in the cellular immune system and which are caused by certain retroviruses. In Aids during the later phase almost always malignant carcinomas or sarcomas occur, such as e.g. Kaposi's disease.
At present no specific therapy for Aids is known. Treatment is still limited at combating to the maximum extent the life-threatening infections and neoplasms. Use is made of different antiviral substances, such as e.g. AZT (azidodeoxythymidine) or stimulators of the immune system, such as e.g. interferons or interleukins.
There is consequently a great need for a medicament making it possible to control, reduce or inhibit malignant tumours in humans and animals, or clinically manifest Aids.
The problem of the invention is consequently to make available such a therapeutic.
-2- According to the invention this is achieved by the use of nicotinamideadenine dinucleotide (NADH), nicotinamide-adenine dinucleotide phosphate (NADPH) or a physiologically compatible salt thereof, use being made of single doses between 1 and 50 mg and preferably 5 and 12.5mg.
The use of such endogenic substances leads to surprising therapeutic successes, without side effects being detected or expected. It is admittedly known that NADH can be successfully used in the treatment of Parkinson's disease (EP-A 89 730 051.3) or depressions (not previously published P 41 00 361.6). The completely surprising finding that these substances can be used in the above-indicated doses in an extremely successful manner in the treatment of malignant tumours or Aids, has resulted from the clinical findings described in detail hereinafter. It has been able to prove that NADH and NADPH or physiologically compatible salts thereof inhibit metastasis formation or bring about remissions thereof and that these substances improve the cellular immune reactions and therefore lead to a regression of clinical Aids symptoms.
Case Descriptions Case 1: Female, aged 63, August 1989 operation for invasive duct carcinoma. One year later multiple liver and bone metastases detected. Four therapy cycles, according to the CMF diagram, further increase of liver and bone metastases. Pain only reduceable with the strongest analgesics. Since January 1991 NADH, initially three times a week 12.5 mg, intravenously and then after four weeks parenteral therapy change to NADH orally, 5 mg every other day. April 1991 radiological detection of metastasis regression, some foci greatly reduced in size and some completely disappeared. Continuation of oral NADH therapy, check 1991, CT scanning reveals further marked regression of liver metastases and bone metastases virtually undetectable. Patient free from pain and no longer requires analgesics.
-3- Case 2: Male, aged 59, colon carcinoma three years earlier, 1990 sonographic and radiological detection of multiple liver metastases of cherry to plum size. Two chemotherapy cycles, Myleran or Endoxan unsuccessful, liver foci increase in size.
December 1990 start of therapy with NADH, initially 12.5mg intravenously three times a week and after four weeks change of therapy to NADH orally, 5 mg, every other day. March 1991 sonographic detection of reduced liver foci size. June 1991 check by CT scanning and sonography reveals an almost complete disappearance of the metastases in tht liver. Subjectively the Patient feels extremely well.
Case 3: Female, aged 52, three years earlier quadrantectomy due to invasive scirrhous carcinoma, January 1990 vertebral metastases detected, April 1990 liver metastases discovered by ultrasonics. Therapy with Novaldex leads to no regression of the metastases. Also no response to a therapy cycle according to the CMF diagram. November 1990 intravenous administration of NADH 12.5 mg every other day. After four weeks change to NADH orally, 5 mg, every other day. Two months after the start of NADH therapy clear regression of liver metastases, as well as disappearance/reduction of vertebral metastases. Check in June 1991 reveals complete regression of bone metastases. Liver metastases greatly reduced or Sfoci no longer detectable.
Case 4: Male, aged 66, February 1990 parvicellular bronchial carcinoma diagnosed, multiple foci in both pulmonary lobes, cytostatic therapy with methotrexate andEndoxan leads to no remission.
October 1990 administration of NADPH parenterally (10 mg intravenously) every other day. Radiographic check in 1991 reveals the remission of the new plastic foci both as regards number and size. Continuation of NADPH therapy, 10 mg intravenously every other day. Check in May 1991 by CT scanning confirms a further reduction of tumour foci in both pulmonary lobes.
-4- Case 5: Male, aged 42, HIV positive, Western Plot positive, since November 1989 clinically manifest Aids with development of Kaposi's disease. Therapy with AZT: stabilization of sarcoma growth for three months, but then despite continued AZT therapy occurrence o new additional sarcoma foci, which had to be operatively removed. Six weeks later reappearance of tumour tissue in the operation area, but also in alternate points-continuation of AZT therapy. Since December 1990 NADH administration; first phase 12.5 mg intravenously every other day, change after four weeks to NADH orally, 5 mg daily.
After eight weeks clear remission of the regenerated tumours.
Check after four months reveals no new growth in the treatment interval, almost complete regression of the sarcoma residue.
Case 6: Male, aged 28, since the end of 1989 clinical symptoms of Aids, recurrent infections, pneumonia, herpetic and fungal infections. HIV positive, Western Plot positive, since mid- 1990 under AZT therapy, no significant improvement in condition during six months administration. Since February 1991 therapy with NADPH, 10 mg intravenously, every other day, infections stopped, at present no pneumonia or fungal infections, laboratory examinations reveal decrease of T-suppressor cells, increase in the ratio of T4 and T8 cells, cellular immune status much better. HIV and Western Plot still positive.
The features of the invention disclosed in the above description and in the claims, both individually and in random combination, can be essential to the realization of the different embodiments of the invention.

Claims (2)

1. A method of treatment of cancer or AIDS comprising administering to a patient requiring such treatment an effective amount of nicotinamide-adenine dinucleotide (NADH), nicotinamide-adenine dinucleotide phosphate (NADPH) or a physiologically compatible salt thereof.
2. A method as claimed in claim 1 wherein single doses of 1 to 50 mg are administered to said patient. A method as claimed in claim 2 wherein singles doses of 5 to 12.5 mg are administered to said patient. DATED this 8th day of August, 1994 UNIV.-PROF. DDR. JORG BIRKMAYER o WATERMARK PATENT TRADEMARK ATTORNEYS THE ATRIUM 290 BURWOOD ROAD HAWTHORN VICTORIA 3122 AUSTRALIA DOC 034 AU2125392.WPC. DBM/KJS:KP I II -6- ABSTRACT Use of nicotillamideadenine dinucle0tide (NADH), nifotinamideaden~ine dinucleotide phosphate (NADPH) or a phgsiologically compatible salt thereof for the treatment of cancer or AIDS, r I r r r r s r to cc a rc i D
AU21253/92A 1991-08-26 1992-08-25 Medicament against cancer and AIDS Ceased AU653619B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE4128625A DE4128625A1 (en) 1991-08-26 1991-08-26 MEDICINE AGAINST CANCER AND AIDS
DE4128625 1991-08-26

Publications (2)

Publication Number Publication Date
AU2125392A AU2125392A (en) 1993-03-04
AU653619B2 true AU653619B2 (en) 1994-10-06

Family

ID=6439356

Family Applications (1)

Application Number Title Priority Date Filing Date
AU21253/92A Ceased AU653619B2 (en) 1991-08-26 1992-08-25 Medicament against cancer and AIDS

Country Status (13)

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EP (1) EP0534097B1 (en)
JP (1) JP3493202B2 (en)
AT (1) ATE150313T1 (en)
AU (1) AU653619B2 (en)
BR (1) BR9203302A (en)
CA (1) CA2072484C (en)
DE (2) DE4128625A1 (en)
DK (1) DK0534097T3 (en)
ES (1) ES2099772T3 (en)
GR (1) GR3023191T3 (en)
HU (1) HUT61895A (en)
NO (1) NO300915B1 (en)
ZA (1) ZA924902B (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1999012951A1 (en) * 1997-09-11 1999-03-18 Oxigene, Inc. Uses of nicotinamide adenine dinucleotide and its analogs for treatment of malignant and infectious diseases
US20040126751A1 (en) * 2002-12-27 2004-07-01 Birkmayer Jorg G.D. Method of prolonging the life-span of living cells using NADH, NADPH and ADP-ribose

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1162938B (en) * 1983-08-26 1987-04-01 Dino Spisni COMPOSITION FOR THE TREATMENT OF MALIGNANT CANCERS, IN PARTICULAR ON ANIMALS
EP0331620B1 (en) * 1988-03-01 1993-08-11 Birkmayer, Walther, Prof. Dr. Agent for the treatment of parkinson's disease

Also Published As

Publication number Publication date
ZA924902B (en) 1993-04-28
NO923324L (en) 1993-03-01
HUT61895A (en) 1993-03-29
EP0534097A3 (en) 1993-07-14
ATE150313T1 (en) 1997-04-15
JPH072678A (en) 1995-01-06
AU2125392A (en) 1993-03-04
DE59208223D1 (en) 1997-04-24
NO300915B1 (en) 1997-08-18
EP0534097A2 (en) 1993-03-31
CA2072484C (en) 2002-02-26
BR9203302A (en) 1993-03-30
JP3493202B2 (en) 2004-02-03
NO923324D0 (en) 1992-08-25
DE4128625A1 (en) 1993-04-08
GR3023191T3 (en) 1997-07-30
DE4128625C2 (en) 1993-08-12
DK0534097T3 (en) 1997-09-22
EP0534097B1 (en) 1997-03-19
CA2072484A1 (en) 1993-02-27
ES2099772T3 (en) 1997-06-01

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